TKTL1 and cancer: To address this challenge, a synthetic macrocyclic peptide (aMD4)‐conjugated cantilever (Figure 5B) was used for HS‐AFM nanoimaging for rapid, single‐molecule recognition imaging of the human tyrosine kinase hepatocyte growth factor (hMET).[221] The results of this study suggest that HS‐AFM could be used as nanoplatform for TKR inhibitors screening and as a molecular diagnostic tool for precise detection of TKR expression and dynamics on the surface of cancer cells.