SAHA‐CDDP‐coupled supramolecular conjugates self‐assembled into nanomicelles, which preferentially accumulated in tumor sites through the EPR effect and further showed remarkable therapeutic efficacy on cisplatin‐resistant NSCLC tumors.[103] The low sensitivity of most patients with advanced gastric cancer to 5‐fluorouridine (5‐FU) can be attributed to the hypermethylation of transcription factor AP‐2 epsilon (TFAP2E). Here, TFAP2E is linked to non-small cell lung carcinoma.