Treatment‐related AEs included (n of six patients): fatigue (3), anemia (3), constipation (2), bruising (2), hypertension (2), dizziness (1), neutropenia (1), thrombocytopenia (2), elevated ALT (2), lymphocytosis (1), hyponatremia (1), headaches (1), elevated AST (1), ankle edema (1), arthralgia (1), dysgeusia (1), and grade 2 protracted thrombocytopenia resulting in a DLT (1). The gene discussed is GPT; the disease is Thrombocytopenia.