GPT and neutropenia: In the 750-mg BID group (n = 4), the most frequently reported (≥75%) all-causality treatment-emergent AEs (TEAEs) were nausea and fatigue (n = 4 each [100.0%]) and leukopenia, neutropenia, constipation, vomiting, ALT increase, alopecia, and rash (n = 3 each [75.0%]) (Table 2).