BPTF (Bromodomain and PHD Finger Transcription Factor/FALZ) has been linked to various cancers including bladder,36 colorectal,37 melanoma,38 and leukemia.39 BPTF has been predicted to be a highly druggable target.28 Until recently no known inhibitors of BPTF had been available to interrogate its role in the onset and progression of cancer. This evidence concerns the gene BPTF and cancer.